BDBM372987 US10597366, Compound 34::US9896418, Compound 34

SMILES Cc1c(C#N)c(Oc2cc(F)cc(F)c2)ccc1S(=O)(=O)C(F)F

InChI Key InChIKey=DQGRVLYEGDANML-UHFFFAOYSA-N

Data  1 IC50  3 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 372987   

TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Peloton Therapeutics

US Patent
LigandPNGBDBM372987(US10597366, Compound 34 | US9896418, Compound 34)
Affinity DataIC50: <5nMAssay Description:HIF-2a: The total assay volume was about 100 uL in the following configuration: 2 uL compound in 100% DMSO, 88 uL buffer with protein and probe and 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent